|
| [[Reseptor histamin H1|H<sub>1</sub>]] || 9.6–16 || Manusia || <ref name="pmid">{{cite journal | vauthors = Ghoneim OM, Legere JA, Golbraikh A, Tropsha A, Booth RG | title = Novel ligands for the human histamine H1 receptor: synthesis, pharmacology, and comparative molecular field analysis studies of 2-dimethylamino-5-(6)-phenyl-1,2,3,4-tetrahydronaphthalenes | journal = Bioorganic & Medicinal Chemistry | volume = 14 | issue = 19 | pages = 6640–58 | date = October 2006 | pmid = 16782354| doi = 10.1016/j.bmc.2006.05.077 }}</ref><ref name="pmid23357028" />
|-
| [[HistamineReseptor H2histamin receptorH2|H<sub>2</sub>]] || >100,000 || [[Canidae|Canine]] || <ref name="pmid1703298">{{cite journal | vauthors = Gantz I, Schäffer M, DelValle J, Logsdon C, Campbell V, Uhler M, Yamada T | title = Molecular cloning of a gene encoding the histamine H2 receptor | journal = Proc. Natl. Acad. Sci. U.S.A. | volume = 88 | issue = 2 | pages = 429–33 | year = 1991 | pmid = 1703298 | pmc = 50824 | doi = 10.1073/pnas.88.2.429| bibcode = 1991PNAS...88..429G | doi-access = free }}</ref>
|-
| [[HistamineReseptor H3histamin receptorH3|H<sub>3</sub>]] || >10,000 || HumanManusia || <ref name="pmid23357028" /><ref name="pmid10347254">{{cite journal | vauthors = Lovenberg TW, Roland BL, Wilson SJ, Jiang X, Pyati J, Huvar A, Jackson MR, Erlander MG | title = Cloning and functional expression of the human histamine H3 receptor | journal = Molecular Pharmacology | volume = 55 | issue = 6 | pages = 1101–7 | date = June 1999 | pmid = 10347254 | doi = 10.1124/mol.55.6.1101| s2cid = 25542667 }}</ref><ref name="pmid11179434">{{cite journal | vauthors = Liu C, Ma X, Jiang X, Wilson SJ, Hofstra CL, Blevitt J, Pyati J, Li X, Chai W, Carruthers N, Lovenberg TW | title = Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow | journal = Molecular Pharmacology | volume = 59 | issue = 3 | pages = 420–6 | date = March 2001 | pmid = 11179434 | doi = 10.1124/mol.59.3.420 | s2cid = 123619 }}</ref>
|-
| [[HistamineReseptor H4histamin receptorH4|H<sub>4</sub>]] || >10,000 || HumanManusia || <ref name="pmid11179434" />
|-
| [[MuscarinicReseptor acetylcholineasetilkolin receptormuskarinik M1|M<sub>1</sub>]] || 80–100 || HumanManusia || <ref name="pmid1346637">{{cite journal | vauthors = Bolden C, Cusack B, Richelson E | title = Antagonism by antimuscarinic and neuroleptic compounds at the five cloned human muscarinic cholinergic receptors expressed in Chinese hamster ovary cells | journal = The Journal of Pharmacology and Experimental Therapeutics | volume = 260 | issue = 2 | pages = 576–80 | date = February 1992 | pmid = 1346637 }}</ref><ref name="pmid23357028" />
|-
| [[MuscarinicReseptor acetylcholineasetilkolin receptormuskarinik M2|M<sub>2</sub>]] || 120–490 || HumanManusia || <ref name="pmid1346637" /><ref name="pmid23357028" />
|-
| [[MuscarinicReseptor acetylcholineasetilkolin receptormuskarinik M3|M<sub>3</sub>]] || 84–229 || Human || <ref name="pmid1346637" /><ref name="pmid23357028" />
|-
| [[MuscarinicReseptor acetylcholineasetilkolin receptormuskarinik M4|M<sub>4</sub>]] || 53–112 || HumanManusia || <ref name="pmid1346637" /><ref name="pmid23357028" />
|-
| [[MuscarinicReseptor acetylcholineasetilkolin receptormuskarinik M5|M<sub>5</sub>]] || 30–260 || HumanManusia || <ref name="pmid1346637" /><ref name="pmid23357028" />
|-
| {{abbrlink|VGSC|Voltage-dependentSaluran sodiumnatrium channelyang bergantung pada tegangan}} || 48,000–86,000 || RatTikus besar || <ref name="pmid11036158" />
|-
| {{abbrlink|hERG|HumanGen EtherTerkait Eter-à-go-go-Related GeneManusia}} || 27,100 ({{abbrlink|IC<sub>50</sub>|Half-maximal inhibitory concentration}}) || HumanManusia || <ref name="pmid8641472">{{cite journal | vauthors = Suessbrich H, Waldegger S, Lang F, Busch AE | title = Blockade of HERG channels expressed in Xenopus oocytes by the histamine receptor antagonists terfenadine and astemizole | journal = FEBS Letters | volume = 385 | issue = 1–2 | pages = 77–80 | date = April 1996 | pmid = 8641472 | doi = 10.1016/0014-5793(96)00355-9 | s2cid = 40355762 | doi-access = free }}</ref>
|- class="sortbottom"
| colspan="4" style="width: 1px;" | ValuesNilainya areadalah K<sub>i</sub> (nM), unlesskecuali otherwisedinyatakan notedlain. TheSemakin smallerkecil the valuenilainya, the moresemakin stronglykuat theobat drugtersebut bindsberikatan todengan thesitus sitetersebut.
|}
| 